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Microdialysis in Drug Development / edited by Markus Müller.

SpringerLink Books Biomedical and Life Sciences 2013 Available online

View online
Format:
Book
Contributor:
Müller, Markus, 1967 August 23- editor.
SpringerLink (Online service)
Series:
Biomedical and Life Sciences (Springer-11642)
AAPS advances in the pharmaceutical sciences series 2210-7371 ; 4.
AAPS Advances in the Pharmaceutical Sciences Series, 2210-7371 ; 4
Language:
English
Subjects (All):
Pharmaceutical technology.
Medicine.
Pharmaceutical Sciences/Technology.
Biomedicine, general.
Local Subjects:
Pharmaceutical Sciences/Technology.
Biomedicine, general.
Physical Description:
1 online resource (XII, 340 pages).
Edition:
First edition 2013.
Contained In:
Springer eBooks
Place of Publication:
New York, NY : Springer New York : Imprint: Springer, 2013.
System Details:
text file PDF
Summary:
In vivo target site concentrations are probably the most important determinant of drug effects. Traditionally, linking drug concentrations to drug effects has been accomplished by modelling blood-derived data, mostly because a direct quantification of tissue concentrations has been beyond technical reach. Today, a direct measurement of target site concentrations is possible by employing microdialysis or complementary approaches such as imaging technologies. Microdialysis, initially conceived in the 1970ies, has become a standard tool in drug development. This comprehensive overview of current microdialysis technology covers general and disease-specific aspects of microdialysis by international experts in the field. It provides useful information for colleagues in academia and industry who are interested PK-PD aspects of drug development.
Contents:
Introduction to the Microdialysis Technology
Recovery and Calibration Techniques: Toward Quantitative Microdialysis
Analytical Considerations for Microdialysis Sampling
Regulatory Aspects of Microdialysis: A United States Food and Drug Administration Perspective
Microdialysis in CNS PKPD Research: Unraveling Unbound Concentrations
Microdialysis in Antibiotic Research
Skin and Transdermal Drug Delivery: Advantages and Challenges
Translational Approaches For Predicting CNS Drug Effects Using Microdialysis
Extracellular Amyloid-β Protein Dynamics in Alzheimer's Disease
Microdialysis in Pain Research
Microdialysis in Ocular Drug Development
Microdialysis in Metabolic Research
High Molecular Weight Targets and Treatments Using Microdialysis
Complementary Techniques - Positron Emission Tomography
Open Flow Microperfusion: An Alternative Method to Microdialysis?
Microdialysis in Internal Organs and Tumors.
Other Format:
Printed edition:
ISBN:
978-1-4614-4815-0
9781461448150
Access Restriction:
Restricted for use by site license.

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